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Carbutamide AHFS /Drugs.com International Drug Names Routes of administration Oral ATC code
4-amino-N -(butylcarbamoyl)benzenesulfonamide
CAS Number PubChem CID ChemSpider UNII ChEMBL CompTox Dashboard (EPA ) ECHA InfoCard 100.005.841 Formula C 11 H 17 N 3 O 3 S Molar mass 271.33 g·mol−1 3D model (JSmol )
O=S(=O)(c1ccc(N)cc1)NC(=O)NCCCC
InChI=1S/C11H17N3O3S/c1-2-3-8-13-11(15)14-18(16,17)10-6-4-9(12)5-7-10/h4-7H,2-3,8,12H2,1H3,(H2,13,14,15)
N Key:VDTNNGKXZGSZIP-UHFFFAOYSA-N
N
N Y (what is this?)
Carbutamide (brand name Glucidoral ) is an anti-diabetic drug of the sulfonylurea class, developed by Servier .
It is classified as first-generation.[1]
It was patented in 1953 and approved for medical use in 1956.[2]
See also [ ]
Hellmuth Kleinsorge (1920-2001) German medical doctor
References [ ]
^ Ballagi-Pordány G, Köszeghy A, Koltai MZ, Aranyi Z, Pogátsa G (January 1990). "Divergent cardiac effects of the first and second generation hypoglycemic sulfonylurea compounds". Diabetes Res. Clin. Pract . 8 (2): 109–14. doi :10.1016/0168-8227(90)90020-T . PMID 2106423 .
^ Fischer, Jnos; Ganellin, C. Robin (2006). Analogue-based Drug Discovery . John Wiley & Sons. p. 449. ISBN 9783527607495 .
Oral
diabetes medication ,
insulins and
insulin analogs , and other drugs used in diabetes (
A10 )
Insulins /insulin analogs
fast-acting short-acting long-acting
Insulin detemir #
Insulin glargine # (+lixisenatide )
NPH insulin
Lente insulin ‡
Ultralente insulin ‡
ultra-long-acting inhalable
# WHO-EM
‡ Withdrawn from market
Clinical trials :
† Phase III
§ Never to phase III
Non-insulins
Insulin sensitizers
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Secretagogues
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Sulfonylureas Meglitinides /"glinides"
GLP-1/GIP receptor agonists DPP-4 inhibitors /"gliptins" FFAR1 agonists
Other
Combinations
# WHO-EM
‡ Withdrawn from market
Clinical trials :
† Phase III
§ Never to phase III
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See also: Receptor/signaling modulators • Transient receptor potential channel modulators
Categories :
Potassium channel blockers Benzenesulfonylureas Anilines Gastrointestinal system drug stubs Hidden categories:
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