Fluetizolam
From Wikipedia, the free encyclopedia
Not to be confused with Flutazolam.
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Formula | C17H15FN4S |
Molar mass | 326.39 g·mol−1 |
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Fluetizolam (2-ethyl-4-(2-fluorophenyl)-9-methyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine) is a thienotriazolodiazepine derivative with potent sedative and anxiolytic effects, which has been sold as a designer drug.[1][2]
See also[]
- Brotizolam
- Clotiazepam
- Flualprazolam
- Flubrotizolam
- Fluclotizolam
- Etizolam
- Ro09-9212
References[]
- ^ EP 0776892, Kitajima H, Ehara S, Sato H, Moriwaki M, Onishi K, "Thienylazole compound and thienotriazolodiazepine compound.", issued 4 June 1997, assigned to Yoshitomi Pharmaceutical
- ^ Catalani V, Botha M, Corkery JM, Guirguis A, Vento A, Scherbaum N, et al. (July 2021). "The Psychonauts' Benzodiazepines; Quantitative Structure-Activity Relationship (QSAR) Analysis and Docking Prediction of Their Biological Activity". Pharmaceuticals (Basel, Switzerland). 14 (8): 720. doi:10.3390/ph14080720. PMC 8398354. PMID 34451817.
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1,4-Benzodiazepines |
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1,5-Benzodiazepines |
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2,3-Benzodiazepines* |
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Triazolobenzodiazepines |
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Imidazobenzodiazepines |
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Oxazolobenzodiazepines |
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Thienodiazepines | |
Thienotriazolodiazepines |
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Thienobenzodiazepines* | |
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Pyridotriazolodiazepines |
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Pyrazolodiazepines | |
Pyrrolodiazepines | |
Tetrahydroisoquinobenzodiazepines | |
Pyrrolobenzodiazepines* |
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Benzodiazepine prodrugs |
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* atypical activity profile (not GABAA receptor ligands) |
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Imidazoles |
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Kava constituents |
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Nonbenzodiazepines |
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Others/unsorted |
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See also: Receptor/signaling modulators • GABA receptor modulators • GABA metabolism/transport modulators |
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